SCHEMBL14748463

SCHEMBL14748463

CCOC(=O)COc1cc(Oc2ccc3c(c2)COB3)ccc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.47
AR P10275 1/20 0.39
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
PDE4A P27815 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 4/20 0.36
HPGD P15428 3/20 0.36
MAPT P10636 3/20 0.36
GLA P06280 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
NTSR1 P30989 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748445 0.88 PDE4B (0.44) PDE4BARNPSR1MEN1KMT2A
SCHEMBL19622210 0.84 PDE4B (0.44) PDE4BARPDE4APDE4CPDE4D
SCHEMBL8007244 0.83 PDE4B (0.42) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748447 0.80 HPGD (0.42) PDE4BNPSR1GAAMEN1KMT2A
SCHEMBL2530250 0.80 PDE4B (0.72) PDE4BPDE4APDE4CPDE4D
SCHEMBL19622201 0.80 PDE4B (0.48) PDE4BARGAAPDE4APDE4C
SCHEMBL14748366 0.76 PDE4B (0.42) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748448 0.75 PDE4B (0.41) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748450 0.74 PDE4B (0.44) PDE4BARPDE4APDE4CPDE4D
SCHEMBL14748429 0.74 PTGS2 (0.43) PDE4BGAAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed