SCHEMBL14764693

SCHEMBL14764693

Cc1ccc2nc(C)c3nnc(-c4cccc(Cl)c4Cl)n3c2c1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 19/20 0.76
PDE10A Q9Y233 16/20 0.76
ESR2 Q92731 1/20 0.56
PDE4D Q08499 1/20 0.56
PDE11A Q9HCR9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14765006 0.90 PDE2A (0.81) PDE2APDE10AESR2PDE4DPDE11A
SCHEMBL14361830 0.88 PDE2A (0.83) PDE2APDE10AESR2PDE4DPDE11A
SCHEMBL14764992 0.86 PDE2A (0.63) PDE2APDE10A
SCHEMBL12502574 0.86 PDE2A (1.00) PDE2APDE10APDE4DPDE11A
SCHEMBL12502753 0.85 PDE2A (1.00) PDE2APDE10A
SCHEMBL12502536 0.80 PDE2A (1.00) PDE2APDE10AESR2PDE4DPDE11A
SCHEMBL14764901 0.80 PDE2A (0.78) PDE2APDE10AESR2PDE4DPDE11A
SCHEMBL3327430 0.80 PDE2A (0.60) PDE2APDE10APDE4D
SCHEMBL3327439 0.79 PDE2A (0.68) PDE2APDE10A
SCHEMBL12503036 0.78 PDE2A (1.00) PDE2APDE10APDE4DPDE11A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO claimed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed