SCHEMBL14764722

SCHEMBL14764722

Cc1nc2c(Br)cccc2nc1Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
TDP1 Q9NUW8 1/20 0.40
PDPK1 O15530 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
BACE1 P56817 2/20 0.35
NQO2 P16083 6/20 0.35
ENPP3 O14638 1/20 0.35
ENPP1 P22413 1/20 0.35
PKMYT1 Q99640 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
PRNP P04156 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764386 0.93 ALDH1A1 (0.42) ALDH1A1TDP1PDPK1NR1H2NR1H3
SCHEMBL30217825 0.93 ALDH1A1 (0.42) ALDH1A1TDP1PDPK1NR1H2NR1H3
SCHEMBL15228704 0.84 TDP1 (0.52) ALDH1A1TDP1PDPK1BACE1NQO2
SCHEMBL30217623 0.84 MAPT (0.44) ALDH1A1TDP1BACE1NQO2PKMYT1
SCHEMBL2513088 0.84 MAPT (0.44) ALDH1A1TDP1BACE1NQO2PKMYT1
SCHEMBL2318402 0.81 NR1H2 (0.46) TDP1L3MBTL1NR1H2NR1H3PIM1
SCHEMBL14764520 0.81 MAPT (0.44) ALDH1A1TDP1L3MBTL1PIM1PIM2
SCHEMBL27763044 0.81 TDP1 (0.41) ALDH1A1TDP1BACE1NQO2PKMYT1
SCHEMBL13313310 0.78 ACHE (0.61) ALDH1A1TDP1L3MBTL1PIM1PIM2
SCHEMBL14764585 0.78 TDP1 (0.40) ALDH1A1TDP1L3MBTL1NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed