SCHEMBL14765153

SCHEMBL14765153

Cc1nc2cccc(F)c2[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.53
DAO P14920 3/20 0.46
DDO Q99489 1/20 0.46
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
TNKS2 Q9H2K2 2/20 0.39
FEN1 P39748 1/20 0.38
TNKS O95271 1/20 0.38
LMNA P02545 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
TYMS P04818 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10285824 0.82 PARP1 (0.50) PARP1DAODDOTNKS2TYMS
SCHEMBL4172152 0.79 PARP1 (0.53) PARP1DAOCA12CA9TNKS2
SCHEMBL14764904 0.79 CA12 (0.43) PARP1DAODDOCA12CA9
SCHEMBL30480783 0.79 KDM4E (0.58) PARP1DAODDOCA12CA9
SCHEMBL10251996 0.79 KDM4E (0.41) PARP1LMNAPOLBHCAR1
SCHEMBL10285538 0.79 PARP1 (0.39) PARP1DAODDOTNKS2
SCHEMBL5142221 0.78 PARP1 (0.59) PARP1DAODDOCA12CA9
SCHEMBL31741632 0.78 KDM4E (0.45) PARP1DAODDOCA12CA9
SCHEMBL15231476 0.77 CASP3 (0.37) PARP1DAODDOTNKS2TNKS
SCHEMBL14765103 0.77 NQO2 (0.45) PARP1DAOTNKS2TNKSLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034758-A1 SUBSTITUTED TRIAZOLOPYRAZINES AND USES THEREOF H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed