SCHEMBL14765103

SCHEMBL14765103

COc1cccc2nc(C)c(=O)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 3/20 0.45
ALDH1A1 P00352 3/20 0.44
ELANE P08246 1/20 0.44
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
CDK9 P50750 1/20 0.43
DYRK1A Q13627 1/20 0.43
GUSB P08236 1/20 0.43
KDM4E B2RXH2 3/20 0.42
HPGD P15428 2/20 0.42
DAO P14920 1/20 0.42
TNKS O95271 1/20 0.42
PARP1 P09874 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
POLB P06746 3/20 0.41
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MCL1 Q07820 2/20 0.41
LMNA P02545 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1041136 0.83 PLAUR (0.50) NQO2ALDH1A1PDE3BPDE3ACDK9
SCHEMBL4611131 0.80 ALDH1A1 (0.46) NQO2ALDH1A1ELANEPDE3BPDE3A
SCHEMBL10285824 0.80 PARP1 (0.50) ALDH1A1ELANEPDE3BPDE3AKDM4E
SCHEMBL16052812 0.77 PDE3B (0.43) NQO2PDE3BPDE3AKDM4EKMT2A
SCHEMBL4172152 0.77 PARP1 (0.53) ELANEPDE3BPDE3ACDK9DYRK1A
SCHEMBL14765153 0.77 PARP1 (0.53) DAOTNKSPARP1TNKS2POLB
SCHEMBL14764904 0.77 CA12 (0.43) CDK9DYRK1AGUSBDAOPARP1
SCHEMBL4420447 0.76 NQO2 (0.46) NQO2ALDH1A1PDE3BPDE3ACDK9
SCHEMBL16053154 0.75 PDE3B (0.38) NQO2PDE3BPDE3AKDM4ETNKS
SCHEMBL14764844 0.75 NQO2 (0.44) NQO2ALDH1A1PDE3BPDE3AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014139983-A1 [1,2,4]TRIAZOLO[4,3-A]QUINOXALINES AS DUAL PDE2/PDE10 INHIBITORS H. LUNDBECK A/S (DK) 2014-09-18 WO disclosed
WO-2013034758-A1 SUBSTITUTED TRIAZOLOPYRAZINES AND USES THEREOF H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed