SCHEMBL14765277

SCHEMBL14765277

COC(=O)Cc1cc(C(=O)c2cccs2)sc1-c1ccc(-c2sccc2C(C)C(=O)O)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.39
ALDH1A1 P00352 4/20 0.39
PTGS1 P23219 3/20 0.39
PTGS2 P35354 3/20 0.39
CYP2C9 P11712 2/20 0.39
LMNA P02545 2/20 0.39
KDM4E B2RXH2 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
TP53 P04637 2/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
HSD17B10 Q99714 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 2/20 0.34
POLB P06746 1/20 0.34
NFKB1 P19838 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14645403 0.87 RAB9A (0.45) HPGDALDH1A1PTGS1PTGS2LMNA
SCHEMBL14645236 0.86 RAB9A (0.41) HPGDALDH1A1PTGS1PTGS2LMNA
SCHEMBL14645324 0.76 NPSR1 (0.38) HPGDALDH1A1CYP2C9LMNAKDM4E
SCHEMBL14646189 0.76 ALDH1A1 (0.55) HPGDALDH1A1PTGS1PTGS2CYP2C9
SCHEMBL14645498 0.76 KMT2A (0.49) HPGDALDH1A1PTGS1PTGS2CYP2C9
SCHEMBL14645336 0.74 NPSR1 (0.43) HPGDALDH1A1CYP2C9LMNAKDM4E
SCHEMBL9976580 0.71 KDM4E (0.47) HPGDALDH1A1LMNAKDM4ENPC1
SCHEMBL15695284 0.70 MEN1 (0.41) HPGDALDH1A1CYP2C9LMNARXFP1
SCHEMBL14646181 0.68 KMT2A (0.41) HPGDALDH1A1LMNAKDM4ENPC1
SCHEMBL14645455 0.67 KMT2A (0.34) HPGDALDH1A1KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036196-A1 NOVEL THIOPHENE COMPOUNDS AND METHOD FOR IN VIVO IMAGING BIOCHROMIX AB (SE) 2013-03-14 WO disclosed