SCHEMBL14767414

SCHEMBL14767414

COc1ccc(-c2ccc(-c3ccc(OCCN4CCCC4)c(OC)c3)nc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 9/20 0.56
HTR2C P28335 1/20 0.52
LTA4H P09960 2/20 0.50
HRH3 Q9Y5N1 1/20 0.49
ABCB1 P08183 1/20 0.49
ADORA2A P29274 2/20 0.48
ADORA1 P30542 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12441119 0.90 MCHR1 (0.58) MCHR1HTR2CHRH3
SCHEMBL12441100 0.86 MCHR1 (0.69) MCHR1LTA4HHRH3
SCHEMBL6957842 0.78 MCHR1 (0.70) MCHR1HTR2CLTA4H
SCHEMBL12440363 0.78 MCHR1 (0.57) MCHR1HRH3
SCHEMBL14767433 0.78 SMN1; SMN2 (0.51) MCHR1HTR2CLTA4HHRH3
SCHEMBL12440267 0.77 MCHR1 (0.67) MCHR1LTA4H
SCHEMBL14767429 0.77 MCHR1 (0.46) MCHR1LTA4HHRH3
SCHEMBL12439925 0.77 SMN1; SMN2 (0.56) MCHR1HTR2CHRH3
SCHEMBL12441464 0.77 MCHR1 (0.53) MCHR1HTR2CLTA4H
SCHEMBL7443460 0.76 LTA4H (0.77) MCHR1LTA4HHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-B1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2013-03-13 EP disclosed