SCHEMBL14767743

SCHEMBL14767743

Cc1sc2[nH]c(=O)nc(NN)c2c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 4/20 0.38
ADORA3 P0DMS8 2/20 0.35
CDC7 O00311 1/20 0.35
ROCK2 O75116 1/20 0.35
MAP4K4 O95819 1/20 0.35
PIM1 P11309 1/20 0.35
GSK3B P49841 1/20 0.35
HIPK2 Q9H2X6 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
GAA P10253 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12323392 0.84 MAPK1 (0.42) MAPK1KDM4EADORA3CDC7ROCK2
SCHEMBL641559 0.78 MAPK1 (0.46) MAPK1KDM4EADORA3CDC7ROCK2
Hydrochloric Acid SCHEMBL643220 0.77 MAPK1 (0.45) MAPK1KDM4EADORA3CDC7ROCK2
SCHEMBL1622415 0.72 MAPK1 (0.44) MAPK1KDM4EADORA3CDC7ROCK2
SCHEMBL23607971 0.69 NPC1 (0.33) ADORA3GAAALDH1A1
SCHEMBL12102045 0.68 MAPK1 (0.55) MAPK1KDM4EADORA3CDC7ROCK2
SCHEMBL16428676 0.65 MAPK1 (0.54) MAPK1KDM4EADORA3PIM1GSK3B
SCHEMBL14767736 0.65 ADORA2A (0.46) MAPK1KDM4EGAASMN1; SMN2LMNA
SCHEMBL12322236 0.64 QPCT (0.38) MAPK1CDC7GAKQPCT
SCHEMBL12322232 0.62 MAPK1 (0.31) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2568287-A2 Modulation of chemosensory receptors and ligands associated Senomyx, Inc. (US) 2013-03-13 EP disclosed