SCHEMBL14775717

SCHEMBL14775717

Nc1c(NC(=O)O)cccc1-c1ccsc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.43
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
IDH2 P48735 7/20 0.41
KDR P35968 3/20 0.41
KIT P10721 2/20 0.41
FLT1 P17948 2/20 0.41
HDAC1 Q13547 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GPR35 Q9HC97 1/20 0.40
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
IKBKB O14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3831632 0.86 HCRTR1 (0.49) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL7119865 0.78 G6PD (0.47) KDRKITFLT1MEN1USP2
SCHEMBL3825744 0.76 POLB (0.46) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL15366094 0.73 KCNH2 (0.46) MEN1USP2MAPTALOX15KMT2A
SCHEMBL975555 0.73 KCNH2 (0.56) HDAC1MAPTIKBKBPTPRFPTPN1
SCHEMBL3831610 0.73 P2RY14 (0.46) IDH2GPR35IKBKBPTPRFPTPN1
SCHEMBL3825279 0.73 IDH2 (0.56) IDH2GPR35
SCHEMBL3827067 0.72 IDH2 (0.52) IDH2
SCHEMBL3846891 0.72 IDH2 (0.51) IDH2
SCHEMBL3844021 0.72 IDH2 (0.44) IDH2MAPTGPR35IKBKBPTPRF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-B1 INHIBITORS OF HISTONE DEACETYLASE MERCK SHARP & DOHME (US) 2013-03-20 EP disclosed