SCHEMBL14775752

SCHEMBL14775752

Cc1nn(-c2ccccc2)c2sc(C(=O)NN3CCCCC3)cc12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.71
HPGD P15428 8/20 0.71
NPSR1 Q6W5P4 4/20 0.71
SMN1; SMN2 Q16637 4/20 0.71
LMNA P02545 3/20 0.71
POLB P06746 3/20 0.71
USP2 O75604 1/20 0.71
CREBBP Q92793 1/20 0.71
KDM4E B2RXH2 8/20 0.69
TSHR P16473 3/20 0.69
GLA P06280 1/20 0.69
PKM P14618 1/20 0.69
HTT P42858 4/20 0.67
NPC1 O15118 2/20 0.67
RAB9A P51151 2/20 0.67
HSD17B10 Q99714 3/20 0.64
MAPT P10636 9/20 0.61
TP53 P04637 3/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL852988 0.99 ALDH1A1 (0.69) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL853835 0.83 ALDH1A1 (0.84) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL853430 0.83 KDM4E (0.76) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL14775545 0.83 MAPT (0.73) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL26943212 0.82 KDM4E (0.72) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL853800 0.81 MAPT (0.85) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL853240 0.80 KDM4E (1.00) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL854227 0.80 KDM4E (0.71) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL861861 0.79 HTT (0.57) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA
SCHEMBL852703 0.79 KDM4E (0.71) ALDH1A1HPGDNPSR1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1775298-B1 THIENOPYRAZOLE DERIVATIVE HAVING PDE7 INHIBITORY ACTIVITY DAIICHI SANKYO CO LTD (JP) 2013-03-20 EP claimed