SCHEMBL14775828

SCHEMBL14775828

Cc1cccc(-c2ccccc2)c1C(=O)N1CC[C@@H](Nc2nc3ccccc3[nH]2)C1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.44
HTR2B P41595 4/20 0.42
ITGB3 P05106 4/20 0.42
ITGAV P06756 4/20 0.42
HRH4 Q9H3N8 1/20 0.41
BACE1 P56817 2/20 0.41
BACE2 Q9Y5Z0 1/20 0.41
CCR5 P51681 1/20 0.41
KCNH2 Q12809 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775830 1.00 PDE10A (0.44) PDE10AHTR2BITGB3ITGAVHRH4
SCHEMBL1141655 0.82 CDK4 (0.49) PDE10AHTR2BBACE1BACE2
SCHEMBL1141659 0.82 CDK4 (0.49) PDE10AHTR2BBACE1BACE2
SCHEMBL9690986 0.80 SMN1; SMN2 (0.51) KCNH2SMN1; SMN2
SCHEMBL1826572 0.80 PDE10A (0.43) PDE10ACCR5
SCHEMBL1826569 0.80 PDE10A (0.43) PDE10ACCR5
Hydrochloric Acid SCHEMBL9382986 0.79 SMN1; SMN2 (0.50) KCNH2SMN1; SMN2
SCHEMBL9630086 0.77 NOS2 (0.51) ITGB3ITGAVKCNH2SMN1; SMN2
Hydrochloric Acid SCHEMBL9594900 0.76 NOS2 (0.50) ITGB3ITGAVKCNH2SMN1; SMN2
SCHEMBL8139051 0.76 SMN1; SMN2 (0.53) KCNH2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2318367-B1 PIPERIDINE AND PYRROLIDINE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2013-03-20 EP disclosed