SCHEMBL14775932

SCHEMBL14775932

CN1CCN(C(Cc2ccccc2C(=O)Nc2cc(-c3ccccc3)ccc2N)C(=O)Nc2ccc3ccccc3c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 8/20 0.46
HDAC3 O15379 6/20 0.46
HDAC1 Q13547 8/20 0.44
ABCB1 P08183 2/20 0.41
WDR5 P61964 4/20 0.41
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2685468 0.87 HDAC1 (0.51) HDAC2HDAC3HDAC1
SCHEMBL2687804 0.84 HDAC1 (0.50) HDAC2HDAC3HDAC1
SCHEMBL5547754 0.80 ABCB1 (0.58) HDAC2HDAC3HDAC1ABCB1
SCHEMBL2686378 0.77 HDAC1 (0.54) HDAC2HDAC3HDAC1
SCHEMBL2684600 0.77 HDAC2 (0.61) HDAC2HDAC3HDAC1ABCB1KCNH2
SCHEMBL2686788 0.77 HDAC2 (0.57) HDAC2HDAC3HDAC1
SCHEMBL2686695 0.77 HDAC1 (0.53) HDAC2HDAC3HDAC1
SCHEMBL2685411 0.77 HDAC1 (0.52) HDAC2HDAC3HDAC1ABCB1
SCHEMBL14775934 0.75 ABCB1 (0.40) HDAC2HDAC3HDAC1ABCB1
SCHEMBL2686432 0.75 HDAC1 (0.52) HDAC2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-B1 INHIBITORS OF HISTONE DEACETYLASE MERCK SHARP & DOHME (US) 2013-03-20 EP disclosed