SCHEMBL14775934

SCHEMBL14775934

CN1CCN(C(CN(C(=O)c2ccccc2)c2cc(-c3ccccc3)ccc2N)C(=O)Nc2ccc3ccccc3c2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 5/20 0.40
HDAC3 O15379 3/20 0.37
HDAC2 Q92769 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HDAC1 Q13547 1/20 0.36
PTGES O14684 1/20 0.36
ALOX5 P09917 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2685468 0.77 HDAC1 (0.51) HDAC3HDAC2HDAC1
SCHEMBL2687804 0.76 HDAC1 (0.50) HDAC3HDAC2HDAC1
SCHEMBL5547754 0.72 ABCB1 (0.58) ABCB1HDAC3HDAC2HDAC1
SCHEMBL2684600 0.70 HDAC2 (0.61) ABCB1HDAC3HDAC2HDAC1
SCHEMBL2685411 0.69 HDAC1 (0.52) ABCB1HDAC3HDAC2HDAC1NPC1
SCHEMBL14775594 0.69 RAB9A (0.51) ABCB1NPC1RAB9AMEN1KMT2A
SCHEMBL8230870 0.68 HDAC2 (0.41) ABCB1HDAC3HDAC2HDAC1
SCHEMBL2686788 0.67 HDAC2 (0.57) HDAC3HDAC2HDAC1
SCHEMBL2686378 0.67 HDAC1 (0.54) HDAC3HDAC2HDAC1
SCHEMBL2686695 0.66 HDAC1 (0.53) HDAC3HDAC2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991226-B1 INHIBITORS OF HISTONE DEACETYLASE MERCK SHARP & DOHME (US) 2013-03-20 EP disclosed