SCHEMBL14809228

SCHEMBL14809228

CCCCCCCCC=CCCCCCCCC(=O)OC(OC(=O)CCCCCCCC=CCCCCCCCC)C(C)[N+](C)(C)C.COS(=O)(=O)[O-]

nearest known ligand 0.51

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 1/20 0.51
PRKCA P17252 2/20 0.46
PRKCE Q02156 1/20 0.46
PRKCQ Q04759 1/20 0.46
PRKCD Q05655 1/20 0.46
LMNA P02545 2/20 0.43
CNR2 P34972 2/20 0.43
FAAH O00519 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
CNR1 P21554 1/20 0.43
EPHX2 P34913 1/20 0.43
DAGLA Q9Y4D2 1/20 0.43
FABP3 P05413 2/20 0.43
DGKA P23743 1/20 0.43
LPAR1 Q92633 1/20 0.42
PGR P06401 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADRA2C P18825 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26134552 1.00 SLC6A5 (0.51) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL625049 0.90 SLC6A5 (0.56) SLC6A5PRKCAPRKCEPRKCQPRKCD
Bromide SCHEMBL29051255 0.89 SLC6A5 (0.55) SLC6A5PRKCAPRKCEPRKCQPRKCD
Hydrochloric Acid SCHEMBL25269826 0.89 SLC6A5 (0.55) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL3371269 0.86 SLC6A5 (0.53) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL23925777 0.85 SLC6A5 (0.55) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL22319402 0.84 SLC6A5 (0.54) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL29449493 0.84 SLC6A5 (0.54) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL5824303 0.83 SLC6A5 (0.50) SLC6A5PRKCAPRKCEPRKCQPRKCD
SCHEMBL6740155 0.81 SLC6A5 (0.51) SLC6A5PRKCAPRKCEPRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9289488-B2 Vaccine engineering AC IMMUNE SA (CH) 2016-03-22 US claimed
WO-2024150064-A1 LIPID BINDING PROTEIN MOLECULE THERAPY ABIONYX PHARMA SA (FR) 2024-07-18 WO disclosed
EP-4322746-A1 USE OF LIPID BINDING PROTEIN-BASED COMPLEXES IN ORGAN PRESERVATION SOLUTIONS Abionyx Pharma SA (FR) 2024-02-21 EP disclosed
WO-2023237927-A2 METHODS FOR TREATING HYPERINFLAMMATORY CONDITIONS USING LIPID BINDING PROTEIN -BASED COMPLEXES ABIONYX PHARMA SA (FR) 2023-12-14 WO disclosed
WO-2023237935-A2 METHODS FOR TREATING ACUTE CONDITIONS USING LIPID BINDING PROTEIN-BASED COMPLEXES ABIONYX PHARMA SA (FR) 2023-12-14 WO disclosed
WO-2023194798-A1 METHODS FOR TREATING LEUKOCYTOSIS, ENDOTHELIAL DYSFUNCTION AND CARDITIS USING LIPID BINDING PROTEIN-BASED COMPLEXES ABIONYX PHARMA SA (FR) 2023-10-12 WO disclosed
EP-3668600-A1 CARGOMERS Abionyx Pharma SA (FR) 2020-06-24 EP disclosed
EP-3668549-A1 APOMERS Abionyx Pharma SA (FR) 2020-06-24 EP disclosed
EP-3527220-A1 VACCINE ENGINEERING AC Immune S.A. (CH) 2019-08-21 EP disclosed
WO-2019030575-A1 APOMERS CERENIS THERAPEUTICS HOLDING (FR) 2019-02-14 WO disclosed
WO-2019030574-A1 CARGOMERS CERENIS THERAPEUTICS HOLDING (FR) 2019-02-14 WO disclosed
EP-2758071-B1 VACCINE THERAPY AC IMMUNE SA (CH) 2018-11-28 EP disclosed
US-9289488-B2 Vaccine engineering AC IMMUNE SA (CH) 2016-03-22 US disclosed
US-20140314837-A1 Vaccine Therapy AC IMMUNE SA (CH) 2014-10-23 US disclosed
EP-2758071-A1 VACCINE THERAPY AC Immune S.A. (CH) 2014-07-30 EP disclosed
US-20130287838-A1 VACCINE ENGINEERING AC IMMUNE S.A. (CH) 2013-10-31 US disclosed
WO-2013044147-A1 VACCINE THERAPY AC IMMUNE S.A. (CH) 2013-03-28 WO disclosed