SCHEMBL14816552

SCHEMBL14816552

Cc1cc2c(cc1C1(c3ccc(C(=O)O)cn3)CC1)C(C)(C)C=CC2(C)C

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 16/20 0.80
RXRB P28702 9/20 0.80
RXRG P48443 9/20 0.80
RARB P10826 5/20 0.80
RARG P13631 5/20 0.80
RARA P10276 4/20 0.80
PPARG P37231 2/20 0.80
MEN1 O00255 1/20 0.39
CYP26A1 O43174 1/20 0.39
ABCB11 O95342 1/20 0.39
ESR1 P03372 1/20 0.39
PGR P06401 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD1 P21728 1/20 0.39
TBXA2R P21731 1/20 0.39
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29434832 0.89 RXRA (1.00) RXRARXRBRXRGRARBRARG
SCHEMBL301213 0.89 RXRA (1.00) RXRARXRBRXRGRARBRARG
SCHEMBL29357483 0.89 RXRA (1.00) RXRARXRBRXRGRARBRARG
SCHEMBL20411355 0.82 RXRA (0.78) RXRARXRBRXRGRARBRARG
SCHEMBL16256670 0.82 RXRA (0.53) RXRARXRBRXRGRARBRARG
SCHEMBL13717021 0.81 RXRA (0.78) RXRARXRBRXRGRARBRARG
SCHEMBL13717159 0.81 PPARG (0.54) RXRARXRBRXRGRARBRARG
SCHEMBL6687036 0.80 RXRA (0.71) RXRARXRBRXRGRARBRARG
SCHEMBL13752425 0.79 RXRA (0.82) RXRARXRBRXRGRARBRARG
SCHEMBL19351439 0.79 RXRA (0.66) RXRARXRBRXRGRARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10391093-B2 Therapeutic compounds ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA, ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2019-08-27 US disclosed
US-20170182046-A1 THERAPEUTIC COMPOUNDS Arizona Board of Regents, a body Corporate of the State of Arizona, Acting for and on Behalf of Ariz (US) 2017-06-29 US disclosed
US-9573906-B2 Therapeutic compounds ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2017-02-21 US disclosed
EP-2910549-A1 1,2,3,4-TETRAHYDRO-1,1,4,4-TETRAMETHYLNAPHTHALENE DERIVATIVES USEFUL AS RXR MODULATORS FOR TREATING ALZHEIMER'S DISEASE AND CANCER Arizona Board of Regents, a Body Corporate of the State of Arizona acting for and on behalf of Arizona State University (US) 2015-08-26 EP disclosed
US-20140343079-A1 THERAPEUTIC COMPOUNDS Arizona Board of Regents, A body corporate of the State of Arizona, acting for and on 2014-11-20 US disclosed
US-20140343079-A1 THERAPEUTIC COMPOUNDS Arizona Board of Regents, A body corporate of the State of Arizona, acting for and on 2014-11-20 US disclosed
WO-2013040227-A2 THERAPEUTIC COMPOUNDS ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2013-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10391093-B2 Therapeutic compounds PSEN1, PSEN2, MAPT RXRA 3433/4885RXRB 3366/4885RXRG 2932/4885
US-20170182046-A1 THERAPEUTIC COMPOUNDS PSEN1, PSEN2, MAPT RXRA 3433/4885RXRB 3366/4885RXRG 2932/4885
US-20140343079-A1 THERAPEUTIC COMPOUNDS MAPT, PSEN1, PSEN2 RXRA 3109/4885RXRB 2990/4885RXRG 2381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.