SCHEMBL14830237

SCHEMBL14830237

Cc1ccc(N(C)C(=O)c2sc(NN(C(=O)O)C(=O)O)nc2-c2ccccc2)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 8/20 0.49
GPBAR1 Q8TDU6 3/20 0.43
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 1/20 0.43
NPSR1 Q6W5P4 3/20 0.41
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ADORA3 P0DMS8 3/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
POLB P06746 1/20 0.38
THRB P10828 1/20 0.38
ADORA2A P29274 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14833280 0.90 DHODH (0.45) DHODHGPBAR1CYP2C19CYP3A4NPSR1
SCHEMBL14814993 0.88 DHODH (0.47) DHODHGPBAR1CYP2C19CYP3A4NPSR1
SCHEMBL14814566 0.88 DHODH (0.51) DHODHGPBAR1CYP2C19CYP3A4NPSR1
SCHEMBL14814905 0.70 GPBAR1 (0.45) DHODHGPBAR1CYP2C19CYP3A4LMNA
SCHEMBL14814884 0.69 GPBAR1 (0.44) DHODHGPBAR1CYP2C19CYP3A4LMNA
SCHEMBL14814904 0.69 GPBAR1 (0.43) DHODHGPBAR1CYP2C19CYP3A4LMNA
SCHEMBL11006800 0.67 SMN1; SMN2 (0.53) GPBAR1CYP2C19CYP3A4GAAALDH1A1
SCHEMBL28719395 0.66 SMN1; SMN2 (0.51) DHODHCYP2C19NPSR1HTTLMNA
SCHEMBL16742064 0.66 DHODH (1.00) DHODH
SCHEMBL14814910 0.63 SMN1; SMN2 (0.46) DHODHCYP2C19NPSR1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013049585-A1 ARYLSUBSTITUTED THIAZOLOTRIAZOLES AND THIAZOLOIMIDAZOLES HENGRUI (USA), LTD. (US) 2013-04-04 WO disclosed