SCHEMBL14833280

SCHEMBL14833280

Cc1ccc(N(C)C(=O)c2sc(NN(C(=O)O)C(=O)OC(C)(C)C)nc2-c2ccccc2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 10/20 0.45
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
NPSR1 Q6W5P4 5/20 0.37
LMNA P02545 4/20 0.37
ADORA3 P0DMS8 2/20 0.37
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 1/20 0.36
PAX8 Q06710 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ADORA2B P29275 1/20 0.36
LCK P06239 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14814993 0.97 DHODH (0.47) DHODHCYP2C19CYP3A4GPBAR1NPSR1
SCHEMBL14830237 0.90 DHODH (0.49) DHODHCYP2C19CYP3A4GPBAR1NPSR1
SCHEMBL14814566 0.81 DHODH (0.51) DHODHCYP2C19CYP3A4GPBAR1NPSR1
SCHEMBL14814910 0.76 SMN1; SMN2 (0.46) DHODHCYP2C19NPSR1LMNAADORA3
SCHEMBL14827149 0.75 KMT2A (0.55) DHODHCYP2C19NPSR1LMNAHTT
SCHEMBL14814557 0.73 DHODH (0.63) DHODHCYP2C19NPSR1ALDH1A1MEN1
SCHEMBL6494266 0.70 CHRNA1 (0.43) CYP2C19CYP3A4GPBAR1SMN1; SMN2MAPT
SCHEMBL14814999 0.69 MEN1 (0.51) NPSR1LMNAADORA3HTTSMN1; SMN2
SCHEMBL14108121 0.65 RAB9A (0.41) CYP2C19SMN1; SMN2MAPTMEN1CYP1A2
SCHEMBL14814905 0.65 GPBAR1 (0.45) DHODHCYP2C19CYP3A4GPBAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013049585-A1 ARYLSUBSTITUTED THIAZOLOTRIAZOLES AND THIAZOLOIMIDAZOLES HENGRUI (USA), LTD. (US) 2013-04-04 WO disclosed