SCHEMBL14838567

SCHEMBL14838567

CCOCc1ccc(CNC)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.47
KDM4E B2RXH2 2/20 0.46
MAPT P10636 2/20 0.46
CYP3A4 P08684 1/20 0.46
NCF1 P14598 2/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
THRB P10828 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ADRB2 P07550 1/20 0.38
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.38
HTR7 P34969 1/20 0.36
TSHR P16473 1/20 0.36
CACNA1G O43497 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1I Q9P0X4 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL133476 0.83 TSHR (0.48) KDM4ECYP3A4THRBTDP1TSHR
SCHEMBL18551296 0.79 KDM4E (0.45) LOXL2KDM4EMAPTCYP3A4NCF1
Benzene SCHEMBL28286600 0.78 TSHR (0.58) KDM4EMAPTCYP3A4ALDH1A1TSHR
SCHEMBL18180057 0.78 APP (0.50) CYP3A4THRBALDH1A1TSHRHPGD
SCHEMBL2504209 0.78 KDM4E (0.68) LOXL2KDM4EMAPTCYP3A4NCF1
SCHEMBL13930293 0.77 LOXL2 (0.50) LOXL2KDM4EMAPTCYP3A4NCF1
SCHEMBL8750395 0.77 TP53 (0.43) MAPTTDP1ALDH1A1TSHRMEN1
SCHEMBL1337544 0.77 AGXT (0.43) TSHR
Dimethylamine SCHEMBL27669857 0.76 TSHR (0.61) KDM4EMAPTCYP3A4ALDH1A1TSHR
Hydrochloric Acid SCHEMBL30925271 0.75 KDM4E (0.74) LOXL2KDM4EMAPTCYP3A4NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140378668-A1 Tyrosine Bioconjugation through Aqueous Ene-Like Reactions SCRIPPS RESEARCH INST (US) 2014-12-25 US disclosed
WO-2013049726-A2 PROCESSES FOR MAKING COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140378668-A1 Tyrosine Bioconjugation through Aqueous Ene-Like Reactions TYR, DNPEP, TH LOXL2 1712/4885KDM4E 225/4885MAPT 1928/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.