SCHEMBL14856502

SCHEMBL14856502

C/C(=N/O)c1ccc(Nc2ccc(Cl)cc2C(F)(F)F)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FLT3 P36888 2/20 0.36
KIT P10721 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
USP2 O75604 1/20 0.36
PABPC1 P11940 1/20 0.36
DHODH Q02127 1/20 0.35
KDR P35968 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
CNR2 P34972 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2811620 1.00 RAB9A (0.39) RAB9ACYP1A2CYP2D6CYP2C19GAA
SCHEMBL2811623 1.00 RAB9A (0.39) RAB9ACYP1A2CYP2D6CYP2C19GAA
SCHEMBL2808251 0.88 KIT (0.38) FLT3KITKDM4EDHODHKDR
SCHEMBL2808253 0.88 KIT (0.38) FLT3KITKDM4EDHODHKDR
SCHEMBL185082 0.88 KIT (0.38) FLT3KITKDM4EDHODHKDR
SCHEMBL184859 0.86 OPRM1 (0.37) CYP2D6FLT3KITKDM4EDHODH
SCHEMBL2811511 0.86 OPRM1 (0.37) CYP2D6FLT3KITKDM4EDHODH
SCHEMBL186306 0.86 RAB9A (0.46) RAB9ACYP1A2CYP2D6CYP2C19GAA
SCHEMBL2808003 0.83 KDM4E (0.41) GAATP53MAPTSMN1; SMN2FLT3
SCHEMBL2808006 0.83 KDM4E (0.41) GAATP53MAPTSMN1; SMN2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed