SCHEMBL14856643

SCHEMBL14856643

O=C(NC1(C(=O)NCc2ccc(Nc3ccc(Cl)cc3C(F)(F)F)cn2)CC1)Oc1ccc2[nH]cnc2c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 8/20 0.37
CNR2 P34972 1/20 0.33
P2RY14 Q15391 2/20 0.33
TRPV1 Q8NER1 3/20 0.31
NTRK1 P04629 1/20 0.31
P2RX7 Q99572 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTK2 Q05397 1/20 0.30
FAAH O00519 2/20 0.30
KDR P35968 1/20 0.30
TEK Q02763 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2809567 0.88 POLB (0.38) CDK1CNR2L3MBTL1POLB
SCHEMBL14857251 0.86 CNR2 (0.36) CNR2TRPV1P2RX7L3MBTL1FAAH
SCHEMBL14856723 0.86 CNR2 (0.36) CNR2TRPV1NTRK1P2RX7L3MBTL1
SCHEMBL14856668 0.85 CNR2 (0.36) CNR2TRPV1P2RX7L3MBTL1FAAH
SCHEMBL14856749 0.85 CNR2 (0.35) CNR2TRPV1P2RX7FAAH
SCHEMBL14856721 0.85 CNR2 (0.38) CNR2TRPV1NTRK1P2RX7L3MBTL1
SCHEMBL14856628 0.84 FAAH (0.33) CDK1CNR2TRPV1P2RX7FAAH
SCHEMBL14856551 0.84 CNR2 (0.34) CNR2TRPV1P2RX7L3MBTL1FAAH
SCHEMBL14856623 0.83 CNR2 (0.37) CNR2TRPV1P2RX7PTK2FAAH
SCHEMBL14856808 0.83 CNR2 (0.38) CNR2TRPV1NTRK1P2RX7FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed