SCHEMBL14857043

SCHEMBL14857043

N#Cc1ccc(CN2C[C@@H]3C[C@H]2CO3)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGKZ Q13574 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
CYP19A1 P11511 4/20 0.40
KCNJ1 P48048 1/20 0.40
KCNH2 Q12809 1/20 0.40
TLR7 Q9NYK1 2/20 0.39
PDE1B Q01064 1/20 0.39
CCNC P24863 2/20 0.38
CDK8 P49336 2/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
CCR2 P41597 1/20 0.37
HSD11B1 P28845 2/20 0.37
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
USP2 O75604 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DRD2 P14416 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15324898 0.81 TLR7 (0.43) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL1929059 0.81 JAK2 (0.43) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL15312373 0.81 TLR7 (0.45) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL22425610 0.81 TLR7 (0.43) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL9953021 0.75 KCNJ1 (0.45) JAK2JAK1KCNJ1KCNH2PDE1B
SCHEMBL14857044 0.75 SIRT2 (0.41) CYP19A1TSHRSMN1; SMN2
SCHEMBL15312545 0.74 CYP51A1 (0.40) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL25153282 0.72 LPL (0.43) DGKZJAK2JAK1TLR7PDE1B
SCHEMBL11145753 0.70 CYP19A1 (0.47) CYP19A1KCNJ1KCNH2CCR2CYP11B1
SCHEMBL13162684 0.68 CCNC (0.41) DGKZJAK2JAK1TLR7PDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2579717-A2 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 Merck Sharp & Dohme Corp. (US) 2013-04-17 EP claimed
WO-2011156245-A2 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2011-12-15 WO claimed