SCHEMBL14857136

SCHEMBL14857136

CC(C)c1nccc(-c2ccccc2)c1C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.43
PIM1 P11309 1/20 0.43
BCAT2 O15382 2/20 0.41
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
CDC7 O00311 2/20 0.39
POLB P06746 1/20 0.38
MKNK1 Q9BUB5 2/20 0.37
MKNK2 Q9HBH9 1/20 0.37
IKBKB O14920 2/20 0.37
CHUK O15111 1/20 0.37
IKBKE Q14164 1/20 0.37
PKMYT1 Q99640 1/20 0.37
CHEK2 O96017 1/20 0.37
FYN P06241 1/20 0.36
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR4 P22455 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4560246 0.87 NTRK1 (0.43) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL23199045 0.80 NTRK1 (0.52) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL14917462 0.78 MKNK1 (0.49) NTRK1PIM1BCAT2MEN1GAA
Acetic Acid SCHEMBL27846617 0.77 NTRK1 (0.50) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL25275838 0.76 BCAT2 (0.44) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL28143127 0.76 CDC7 (0.46) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL1533660 0.76 NTRK1 (0.43) NTRK1PIM1BCAT2MEN1GAA
SCHEMBL1591434 0.76 NTRK1 (0.33) NTRK1PIM1CDC7MKNK1MKNK2
SCHEMBL23116461 0.76 SIRT3 (0.41) NTRK1PIM1POLBPKMYT1HSP90AA1
SCHEMBL9215517 0.76 KDM4E (0.39) NTRK1PIM1CDC7HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2579717-A2 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 Merck Sharp & Dohme Corp. (US) 2013-04-17 EP disclosed
WO-2011156245-A2 POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 MERCK SHARP & DOHME CORP. (US) 2011-12-15 WO disclosed