SCHEMBL1485801

SCHEMBL1485801

COC(C(N)=O)=C(C(=O)O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
SRC P12931 1/20 0.44
MAPT P10636 5/20 0.43
POLB P06746 3/20 0.43
TDP1 Q9NUW8 3/20 0.43
CYP2C19 P33261 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP3A4 P08684 2/20 0.43
PARP1 P09874 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
ALDH1A1 P00352 6/20 0.43
LMNA P02545 2/20 0.43
F2 P00734 2/20 0.42
GAA P10253 1/20 0.40
KMT2A Q03164 4/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27589200 0.85 TSHR (0.48) TSHRSRCMAPTPOLBTDP1
SCHEMBL9359710 0.81 MEN1 (0.46) TSHRMAPTPOLBHSD17B10ALDH1A1
SCHEMBL9359702 0.81 MEN1 (0.46) TSHRMAPTPOLBHSD17B10ALDH1A1
SCHEMBL7675491 0.79 TSHR (0.50) TSHRSRCMAPTPOLBTDP1
SCHEMBL27923392 0.77 TSHR (0.52) TSHRSRCMAPTPOLBTDP1
SCHEMBL8975527 0.76 TSHR (0.56) TSHRSRCMAPTPOLBTDP1
SCHEMBL6208814 0.76 TSHR (0.50) TSHRSRCMAPTPOLBTDP1
SCHEMBL937374 0.75 TSHR (0.48) TSHRMAPTPOLBTDP1CYP2C19
SCHEMBL937370 0.75 TSHR (0.48) TSHRMAPTPOLBTDP1CYP2C19
SCHEMBL4405815 0.75 TSHR (0.54) TSHRSRCMAPTTDP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9028787-B2 Preventing or reducing scale in wet-process phosphoric acid production CYTEC TECHNOLOGY CORP. (US) 2015-05-12 US claimed
EP-2688837-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION Cytec Technology Corp. (US) 2014-01-29 EP claimed
US-20120244058-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2012-09-27 US claimed
WO-2012128755-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2012-09-27 WO claimed
EP-2480496-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION Cytec Technology Corporation (US) 2012-08-01 EP claimed
WO-2011038167-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2011-03-31 WO claimed
US-20110076219-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2011-03-31 US claimed
CN-102712476-B Preventing or reducing scale in wet-process phosphoric acid production 塞特克技术公司 2019-03-12 CN disclosed
EP-2480495-B1 PROCESS AND REAGENTS FOR THE INHIBITION OR REDUCTION OF SCALE FORMATION DURING PHOSPHORIC ACID PRODUCTION CYTEC TECH CORPORATION (US) 2018-11-14 EP disclosed
CN-103429528-B The dirt prevented or reduce in Wet-process Phosphoric Acid Production 塞特克技术公司 2016-08-10 CN disclosed
US-9028787-B2 Preventing or reducing scale in wet-process phosphoric acid production CYTEC TECHNOLOGY CORP. (US) 2015-05-12 US disclosed
US-8900539-B2 Preventing or reducing scale in wet-process phosphoric acid production CYTEC TECHNOLOGY CORP. (US) 2014-12-02 US disclosed
EP-2688837-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION Cytec Technology Corp. (US) 2014-01-29 EP disclosed
US-20120244058-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2012-09-27 US disclosed
WO-2012128755-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2012-09-27 WO disclosed
EP-2480496-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION Cytec Technology Corporation (US) 2012-08-01 EP disclosed
WO-2011038167-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2011-03-31 WO disclosed
US-20110076219-A1 PREVENTING OR REDUCING SCALE IN WET-PROCESS PHOSPHORIC ACID PRODUCTION CYTEC TECHNOLOGY CORP. (US) 2011-03-31 US disclosed