SCHEMBL14864458

SCHEMBL14864458

COc1ccc(/C=C/n2c(=O)sc3cc(C)ccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.50
RELA Q04206 3/20 0.45
PADI4 Q9UM07 1/20 0.41
ALOX5 P09917 3/20 0.40
MAPT P10636 3/20 0.40
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
THRB P10828 1/20 0.40
MAOB P27338 2/20 0.39
ADORA2A P29274 1/20 0.39
MAOA P21397 1/20 0.39
AHR P35869 1/20 0.38
TUBB1 Q9H4B7 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ABL1 P00519 1/20 0.38
TTR P02766 1/20 0.38
ESR1 P03372 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1A2 P05177 1/20 0.38
ABCB1 P08183 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13394314 0.84 SMN1; SMN2 (0.45) RELAMAPTTP53SMN1; SMN2MAOB
SCHEMBL3305491 0.83 SMN1; SMN2 (0.54) RELAPADI4MAPTTP53SMN1; SMN2
SCHEMBL3305497 0.83 SMN1; SMN2 (0.54) RELAPADI4MAPTTP53SMN1; SMN2
SCHEMBL1850928 0.82 NFE2L2 (0.50) MAPTMAOBMAOAALDH1A1CYP19A1
SCHEMBL1850926 0.82 NFE2L2 (0.50) MAPTMAOBMAOAALDH1A1CYP19A1
SCHEMBL3306493 0.82 SMN1; SMN2 (0.43) HTR6MAPTTP53SMN1; SMN2AHR
SCHEMBL3306489 0.82 SMN1; SMN2 (0.43) HTR6MAPTTP53SMN1; SMN2AHR
SCHEMBL3307664 0.78 SMN1; SMN2 (0.47) ALOX5MAPTSMN1; SMN2THRBMAOB
SCHEMBL3307658 0.78 SMN1; SMN2 (0.47) ALOX5MAPTSMN1; SMN2THRBMAOB
SCHEMBL13394312 0.76 NFE2L2 (0.51) HTR6RELAALOX5MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8420052-B2 Imaging agents useful for identifying AD pathology SIEMENS MEDICAL SOLUTIONS USA, INC. (US) 2013-04-16 US disclosed