SCHEMBL14865199

SCHEMBL14865199

CC(C(=O)N1CCN[C@H](C)C1)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLD1 Q13393 2/20 0.40
PLD2 O14939 1/20 0.40
BIRC2 Q13490 3/20 0.40
HRH4 Q9H3N8 1/20 0.38
CYP3A4 P08684 2/20 0.34
UGCG Q16739 2/20 0.34
TP53 P04637 1/20 0.33
MDM2 Q00987 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA3 P32297 2/20 0.33
CHRNA4 P43681 2/20 0.33
CHRNB3 Q05901 2/20 0.33
CHRNA6 Q15825 2/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
REN P00797 1/20 0.32
XIAP P98170 2/20 0.31
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14164982 0.82 CHRNB2 (0.48) PLD1PLD2BIRC2HRH4CYP3A4
SCHEMBL26814687 0.82 CHRNB2 (0.48) PLD1PLD2BIRC2HRH4CYP3A4
SCHEMBL14165240 0.82 CHRNB2 (0.48) PLD1PLD2BIRC2HRH4CYP3A4
SCHEMBL30232419 0.80 HPGD (0.44) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL4975517 0.78 PLD1 (0.37) PLD1PLD2BIRC2HRH4CYP3A4
SCHEMBL14397191 0.77 BIRC2 (0.43) PLD1PLD2BIRC2HRH4CYP3A4
SCHEMBL19284233 0.75 BIRC2 (0.44) PLD1PLD2BIRC2HRH4TP53
SCHEMBL28829771 0.75 BIRC2 (0.44) PLD1PLD2BIRC2HRH4TP53
SCHEMBL16501762 0.75 BIRC2 (0.44) PLD1PLD2BIRC2HRH4TP53
Tert-Butyl Formate SCHEMBL28876717 0.75 PLD1 (0.38) PLD1PLD2BIRC2HRH4CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398780-B1 CYCLOPROPYL AMIDE DERIVATIVES TARGETING THE HISTAMINE H3 RECEPTOR ASTRAZENECA AB (SE) 2013-04-17 EP disclosed