SCHEMBL14865374

SCHEMBL14865374

C[C@@]1(C(=O)NCc2ncc(Nc3ccc(Cl)cc3C(F)(F)F)cc2F)CCOC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 11/20 0.39
TP53 P04637 3/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
RAB9A P51151 3/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
P2RX7 Q99572 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
PAX8 Q06710 1/20 0.35
MAPT P10636 2/20 0.35
POLB P06746 1/20 0.35
CNR1 P21554 2/20 0.34
BACE1 P56817 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KIT P10721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2812273 0.88 CNR2 (0.38) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL15455029 0.88 CNR2 (0.38) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL2810858 0.83 CNR2 (0.38) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL14865294 0.83 P2RX7 (0.36) CNR2P2RX7HTT
SCHEMBL186318 0.83 CNR2 (0.37) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL2809124 0.82 CNR2 (0.36) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL2812255 0.82 CNR2 (0.35) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL13129178 0.82 CNR2 (0.37) CNR2TP53CYP1A2RAB9ACYP2D6
SCHEMBL185729 0.82 CNR2 (0.35) CNR2TP53CYP1A2CYP3A4CYP2C9
SCHEMBL2807388 0.82 BDKRB1 (0.39) CNR2TP53CYP1A2RAB9ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed