SCHEMBL14865508

SCHEMBL14865508

CCOC(=O)c1c(C(C)=O)c2ccccc2n1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
KDM4E B2RXH2 5/20 0.58
EGFR P00533 1/20 0.52
SRC P12931 1/20 0.52
KMT2A Q03164 3/20 0.52
PKM P14618 2/20 0.52
GAA P10253 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
TSHR P16473 3/20 0.50
GABRP O00591 1/20 0.50
GABRD O14764 1/20 0.50
GABRA1 P14867 1/20 0.50
GABRB1 P18505 1/20 0.50
GABRG2 P18507 1/20 0.50
GABRB3 P28472 1/20 0.50
GABRA5 P31644 1/20 0.50
GABRA3 P34903 1/20 0.50
GABRA2 P47869 1/20 0.50
GABRB2 P47870 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16110173 0.89 KDM4E (0.58) ALDH1A1KDM4EEGFRSRCKMT2A
SCHEMBL7950698 0.87 ALDH1A1 (0.56) ALDH1A1KDM4EEGFRSRCKMT2A
SCHEMBL16110166 0.86 ALDH1A1 (0.55) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL30639225 0.84 TSHR (0.66) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL7878088 0.84 TSHR (0.66) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL27765520 0.83 KDM4E (0.61) ALDH1A1KDM4EGAATSHRGABRP
SCHEMBL9867870 0.82 ALDH1A1 (0.68) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL23931478 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL1920160 0.81 MAPT (0.62) ALDH1A1KDM4EKMT2APKMGAA
SCHEMBL8689676 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EKMT2APKMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692157-B1 INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE VERTEX PHARMA (US) 2013-04-17 EP disclosed