(S)-Verapamil

(S)-Verapamil

SCHEMBL14874635

COc1ccc(CCN(C)CCC[C@@](C#N)(c2ccc(OC)c(OC)c2)C(C)C)cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CACNA1CCACNA1DCACNA1FCACNA1S

The experimentally established mechanism targets of (S)-Verapamil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C known ✓ Q13936 3/20 1.00
CACNA1F known ✓ O60840 2/20 1.00
CACNA1D known ✓ Q01668 2/20 1.00
CACNA1S known ✓ Q13698 2/20 1.00
ABCB1 P08183 9/20 1.00
CYP3A4 P08684 8/20 1.00
ABCC1 P33527 4/20 1.00
KCNH2 Q12809 3/20 1.00
TSHR P16473 3/20 1.00
LMNA P02545 3/20 1.00
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
CYP2C19 P33261 2/20 1.00
ABCB11 O95342 2/20 1.00
HTR1A P08908 2/20 1.00
ADRA2A P08913 2/20 1.00
DRD2 P14416 2/20 1.00
ADRA2C P18825 2/20 1.00
HTR2A P28223 2/20 1.00
HTR2C P28335 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Verapamil SCHEMBL29450374 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
(S)-Verapamil SCHEMBL29768846 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Dexverapamil SCHEMBL30402443 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Verapamil SCHEMBL29450364 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Verapamil SCHEMBL29064783 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Verapamil SCHEMBL16742 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Dexverapamil SCHEMBL33297 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Dexverapamil SCHEMBL29423253 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Verapamil SCHEMBL1902363 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR
Verapamil SCHEMBL29440902 1.00 ABCB1 (1.00) ABCB1CYP3A4ABCC1KCNH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4314018-A1 METHODS AND COMPOSITIONS FOR HIGH-POTENCY POLYPEPTIDE-BASED PROTEIN INHIBITION Baylor College of Medicine (US) 2024-02-07 EP claimed
US-20230355711-A1 VIMENTIN AND FRAGMENTS OR DERIVATIVES THEREOF FOR CORONAVIRUS TREATMENT AND PREVENTION THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERANS AFFAIRS 2023-11-09 US claimed
US-20230210902-A1 SARS-COV-2-SPECIFIC T CELLS NATIONAL INSTITUTES OF HEALTH 2023-07-06 US claimed
EP-4149496-A1 SARS-COV-2-SPECIFIC T CELLS Board of Regents, The University of Texas System (US) 2023-03-22 EP claimed
US-20220401553-A1 PARAPOXVIRUS FOR CONDITIONING FOR AND TREATMENT OF CORONAVIRUS INFECTIONS AICURIS GMBH & CO. KG (DE) 2022-12-22 US claimed
WO-2022213076-A1 METHODS AND COMPOSITIONS FOR HIGH-POTENCY POLYPEPTIDE-BASED PROTEIN INHIBITION BAYLOR COLLEGE OF MEDICINE (US) 2022-10-06 WO claimed
EP-3906970-B1 PARAPOXVIRUS FOR CONDITIONING AND TREATMENT OF CORONAVIRUS INFECTIONS AICURIS GMBH & CO KG (DE) 2022-07-06 EP claimed
US-20220193204-A1 USES OF A2 DOMAIN OF VON WILLEBRAND FACTOR BAYLOR COLLEGE OF MEDICINE (US) 2022-06-23 US claimed
EP-3969036-A1 USES OF A2 DOMAIN OF VON WILLEBRAND FACTOR Baylor College of Medicine (US) 2022-03-23 EP claimed
US-20150209308-A1 METHODS TO INHIBIT INTRACELLULAR GROWTH OF BACTERIA AND TO TREAT BACTERIA-MEDIATED DISEASES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH 2015-07-30 US claimed
US-9078873-B2 Compositions and methods for preventing cardiac arrhythmia CORMATRIX CARDIOVASCULAR, INC. (US) 2015-07-14 US claimed
US-20150150913-A1 Compositions and Methods for Preventing Cardiac Arrhythmia CORVIVO CARDIOVASCULAR, INC. 2015-06-04 US claimed
WO-2014039011-A1 METHODS TO INHIBIT INTRACELLULAR GROWTH OF BACTERIA AND TO TREAT BACTERIA-MEDIATED DISEASES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-03-13 WO claimed
US-12606631-B2 Antibodies which bind human endothelin receptor a (ETAR) REMD BIOTHERAPEUTICS INC (US) 2026-04-21 US disclosed
EP-4714452-A1 METHODS FOR TREATING SARS COV-2 INFECTIONS Gilead Sciences, Inc. (US) 2026-03-25 EP disclosed
US-20250149121-A1 DETECTION OF PEPTIDE STRUCTURES FOR DIAGNOSING AND TREATING SEPSIS AND COVID VENN BIOSCIENCES CORPORATION 2025-05-08 US disclosed
US-20150073535-A1 Treatment of coronary artery lesions with a scaffold having vessel scaffold interactions that reduce or prevent angina ABBOTT CARDIOVASCULAR SYSTEMS INC. 2015-03-12 US disclosed
WO-2014039011-A1 METHODS TO INHIBIT INTRACELLULAR GROWTH OF BACTERIA AND TO TREAT BACTERIA-MEDIATED DISEASES AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2014-03-13 WO disclosed
US-20130101666-A1 LIPOSOME INCLUDING ELASTIN-LIKE POLYPEPTIDE CONJUGATED TO MOIETY CONTAINING HYDROPHOBIC GROUP, CHEMOSENSITIZER AND ANTICANCER AGENT AND USE THEREOF SAMSUNG ELECTRONICS CO., LTD. (KR) 2013-04-25 US disclosed
EP-2583690-A1 Liposome including elastin-like polypeptide hydrophobic group conjugate, chemosensitizer and anticancer agent and use thereof Samsung Electronics Co., Ltd (KR) 2013-04-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12606631-B2 Antibodies which bind human endothelin receptor a (ETAR) EDNRA, EDNRB, FCGR2A CACNA1C 1226/4885CACNA1F 1118/4885CACNA1D 642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.