SCHEMBL14877482

SCHEMBL14877482

CC1CC(Oc2ccnc3cc(C(F)(F)F)ccc23)CN1C

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.44
NCF1 P14598 1/20 0.44
IDO1 P14902 4/20 0.42
GAK O14976 1/20 0.40
CYP3A4 P08684 1/20 0.36
SCD O00767 4/20 0.36
GRM4 Q14833 1/20 0.35
KDR P35968 2/20 0.35
ACVR1 Q04771 1/20 0.35
CYP8B1 Q9UNU6 1/20 0.35
AAK1 Q2M2I8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8277163 0.84 IDO1 (0.40) ADRB2NCF1IDO1GAKCYP3A4
SCHEMBL14877512 0.83 KMT2A (0.46) ADRB2NCF1IDO1CYP3A4
SCHEMBL14877496 0.82 MET (0.42) GAKKDR
SCHEMBL14877543 0.80 HCRTR1 (0.48) IDO1CYP3A4
SCHEMBL12213692 0.80 IDO1 (0.41) ADRB2NCF1IDO1GAKCYP3A4
SCHEMBL10058159 0.79 IDO1 (0.41) ADRB2NCF1IDO1GAKCYP3A4
SCHEMBL13627379 0.78 IDO1 (0.41) ADRB2NCF1IDO1GAKCYP3A4
SCHEMBL2797692 0.73 GAK (0.64) ADRB2NCF1GAKKDRAAK1
SCHEMBL13409691 0.72 GAK (0.49) ADRB2NCF1IDO1GAKGRM4
SCHEMBL23379637 0.71 ALDH1A1 (0.40) IDO1CYP8B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8426359-B2 Inhibitors of serine proteases, particularly HCV NS3-NS4A protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-23 US disclosed