SCHEMBL14896135

SCHEMBL14896135

COc1ccccc1-c1[c]cncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 2/20 0.43
GAA P10253 2/20 0.43
TP53 P04637 1/20 0.43
NPC1 O15118 1/20 0.43
PDE5A O76074 2/20 0.42
APP P05067 1/20 0.42
KDM4E B2RXH2 2/20 0.41
SLC22A12 Q96S37 1/20 0.41
CYP19A1 P11511 1/20 0.40
HPGD P15428 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
METAP2 P50579 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6639533 0.85 MGAM (0.46) ALDH1A1SMN1; SMN2RAB9AGAATP53
SCHEMBL28056415 0.79 SCN9A (0.41) ALDH1A1KDM4E
SCHEMBL27925023 0.76 GPBAR1 (0.37) ALDH1A1PTGS2
SCHEMBL336434 0.74 APP (0.47) ALDH1A1SMN1; SMN2RAB9AGAATP53
SCHEMBL27958531 0.73 NPC1 (0.39) ALDH1A1RAB9ANPC1KDM4ETDP1
SCHEMBL27473801 0.73 NPC1 (0.39) ALDH1A1SMN1; SMN2RAB9ATP53NPC1
SCHEMBL30141977 0.72 RAB9A (0.61) ALDH1A1SMN1; SMN2RAB9AGAATP53
SCHEMBL4779549 0.72 RAB9A (0.61) ALDH1A1SMN1; SMN2RAB9AGAATP53
Hydrochloric Acid SCHEMBL4778775 0.71 RAB9A (0.59) ALDH1A1SMN1; SMN2RAB9AGAATP53
SCHEMBL1971146 0.70 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2RAB9AGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108699028-B Substituted 4-phenylpyridines as non-systemic TGR5 agonists 阿德利克斯公司 2021-10-22 CN disclosed
WO-2013062887-A1 SUBSTITUTED PYRIDINE DERIVATIVES USEFUL AS GPR131 AGONISTS MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed