SCHEMBL14896367

SCHEMBL14896367

O=[N+]([O-])c1cccc(-n2ccnn2)c1-n1ccnn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 4/20 0.40
TDP1 Q9NUW8 3/20 0.38
PDE10A Q9Y233 1/20 0.37
GPR35 Q9HC97 1/20 0.37
POLB P06746 1/20 0.36
KEAP1 Q14145 1/20 0.36
KMT2A Q03164 2/20 0.36
NOS1 P29475 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MITF O75030 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NCOA1 Q15788 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4457137 0.86 HTT (0.40) NOTUMTDP1KMT2ASMN1; SMN2MAPT
SCHEMBL30721401 0.84 NOTUM (0.45) NOTUMTDP1KMT2ASMN1; SMN2MAPT
SCHEMBL17373622 0.72 NOTUM (0.42) NOTUMKEAP1CYP1A2CYP2C9CYP2C19
SCHEMBL27815199 0.72 LMNA (0.52) NOTUMPOLBKMT2AMAPTHTT
SCHEMBL20766489 0.72 NOTUM (0.41) NOTUMPOLBKEAP1KMT2AMAPT
SCHEMBL31717453 0.72 TSHR (0.49) NOTUMPOLBKMT2ASMN1; SMN2MITF
SCHEMBL17743329 0.72 ALDH1A1 (0.47) NOTUMTDP1KMT2AMAPTHTT
Hydrochloric Acid SCHEMBL23291644 0.71 NOTUM (0.41) NOTUMKEAP1CYP1A2CYP2C9CYP2C19
SCHEMBL17028392 0.71 NOTUM (0.41) NOTUMTDP1POLBKEAP1ALDH1A1
SCHEMBL302445 0.70 MAPK9 (0.41) NOTUMKEAP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2771332-A1 HIV PROTEASE INHIBITORS Merck Canada Inc. (CA) 2014-09-03 EP disclosed
WO-2013059928-A1 HIV PROTEASE INHIBITORS MERCK CANADA INC. (CA) 2013-05-02 WO disclosed