SCHEMBL14899253

SCHEMBL14899253

COc1cccc([C@H]2[C@H](Cn3nnc(CCOO)n3)OC(=O)N2c2ccc(Cl)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HSD11B1 P28845 1/20 0.33
GRM5 P41594 1/20 0.33
GPBAR1 Q8TDU6 2/20 0.33
P2RX3 P56373 1/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
NR1H2 P55055 1/20 0.32
MEN1 O00255 1/20 0.32
CYP2C9 P11712 1/20 0.32
KMT2A Q03164 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TNKS O95271 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3586688 0.92 ALDH1A1 (0.36) ALDH1A1HSD11B1GRM5GPBAR1P2RX3
SCHEMBL13168051 0.91 ALDH1A1 (0.37) ALDH1A1HSD11B1GRM5GPBAR1P2RX3
SCHEMBL15181965 0.88 ALDH1A1 (0.37) ALDH1A1HSD11B1GPBAR1P2RX3CNR1
SCHEMBL3593936 0.88 ALDH1A1 (0.35) ALDH1A1HSD11B1GRM5GPBAR1P2RX3
SCHEMBL3595312 0.86 CHRNA7 (0.39) ALDH1A1
SCHEMBL3585046 0.86 MDM2 (0.38) ALDH1A1CNR1CNR2MEN1CYP2C9
SCHEMBL3579493 0.85 PKM (0.39) ALDH1A1GPBAR1P2RX3SMN1; SMN2MEN1
SCHEMBL3580505 0.84 RECQL (0.43) ALDH1A1GRM5SMN1; SMN2MEN1CYP2C9
SCHEMBL3597651 0.82 CACNA1D (0.42) ALDH1A1GPBAR1P2RX3SMN1; SMN2CYP2C9
SCHEMBL3598128 0.81 MEN1 (0.40) ALDH1A1GRM5SMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8431607-B2 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity IRM LLC, A DELAWARE LIMITED LIABILITY COMPANY (BM) 2013-04-30 US disclosed