SCHEMBL14900002

SCHEMBL14900002

Cc1cc(C(C)(F)F)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CASR P41180 1/20 0.41
ACHE P22303 1/20 0.39
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
ESR1 P03372 1/20 0.37
NR3C1 P04150 1/20 0.35
PDE2A O00408 2/20 0.34
TSHR P16473 3/20 0.33
PTGS2 P35354 2/20 0.33
PTGS1 P23219 1/20 0.33
IDO1 P14902 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
APP P05067 1/20 0.32
DAPK3 O43293 1/20 0.32
NTRK1 P04629 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17506782 0.84 HDAC1 (0.37) HDAC3HDAC1HDAC2HDAC6ACHE
SCHEMBL3949636 0.83 ESR1 (0.54) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL7836049 0.83 TSHR (0.46) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL476625 0.83 PDE2A (0.47) ACHEPDE2AIDO1
SCHEMBL14748164 0.80 ALDH1A1 (0.40) HDAC1HDAC6ESR1PDE2ATSHR
SCHEMBL3950682 0.79 ESR1 (0.43) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL19433290 0.79 CASR (0.40) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL8257902 0.79 CASR (0.46) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL12956711 0.79 CASR (0.40) HDAC3HDAC1HDAC2HDAC6CASR
SCHEMBL24746116 0.79 HSD11B1 (0.46) HDAC3HDAC1HDAC2HDAC6CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414330-B1 Piperidine and piperazine derivatives as autotaxin inhibitors MERCK PATENT GMBH (DE) 2013-05-01 EP disclosed