SCHEMBL1490577

SCHEMBL1490577

COC(=O)c1c(NC(=O)OCc2ccccc2)csc1-c1ccc(Br)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC2 Q92769 3/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ROCK2 O75116 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TACR3 P29371 1/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 1/20 0.39
PTPN1 P18031 1/20 0.39
MGLL Q99685 1/20 0.38
ELANE P08246 3/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490425 0.88 RAB9A (0.48) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490684 0.84 NPC1 (0.52) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490594 0.83 MGLL (0.52) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490651 0.83 NPC1 (0.48) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490619 0.81 NPC1 (0.44) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490433 0.79 NPC1 (0.44) NPC1RAB9ASMN1; SMN2TACR3POLB
SCHEMBL3555247 0.78 NPC1 (0.58) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL12756642 0.78 HDAC3 (0.50) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490217 0.76 NPC1 (0.52) HDAC3HDAC1HDAC2NPC1RAB9A
SCHEMBL1490620 0.74 RAB9A (0.47) HDAC3HDAC1HDAC2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140051711-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2014-02-20 US disclosed
US-8618307-B2 Compounds that modulate intracellular calcium CALCIMEDICA, INC. (US) 2013-12-31 US disclosed
EP-2477982-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2012-07-25 EP disclosed
WO-2011034962-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-03-24 WO disclosed
US-20110065724-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2011-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140051711-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 HDAC3 1653/4885HDAC1 2696/4885HDAC2 2333/4885
US-20110065724-A1 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM ORAI1, SARAF, RYR2 HDAC3 1653/4885HDAC1 2696/4885HDAC2 2333/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.