SCHEMBL14906370

SCHEMBL14906370

FC(F)(F)c1cc(-c2cncn2-c2cnccc2-c2ccc(Cl)cc2)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 10/20 0.40
KLRK1 P26718 2/20 0.37
MICA Q29983 2/20 0.37
RAET1L Q5VY80 2/20 0.37
CYP19A1 P11511 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
HSP90AA1 P07900 2/20 0.34
HSP90AB1 P08238 2/20 0.34
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34
SLC22A12 Q96S37 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14906417 0.91 GPBAR1 (0.36) GPBAR1KLRK1MICARAET1LHSP90AA1
SCHEMBL14906381 0.89 SRC (0.38) GPBAR1KLRK1MICARAET1LHSP90AA1
SCHEMBL14906369 0.89 IDO1 (0.42) GPBAR1CYP19A1
SCHEMBL14906407 0.89 GPBAR1 (0.40) GPBAR1RAB9A
SCHEMBL14906413 0.89 GPBAR1 (0.39) GPBAR1
SCHEMBL14906367 0.89 KLRK1 (0.39) GPBAR1KLRK1MICARAET1LS1PR1
SCHEMBL14906516 0.88 GPBAR1 (0.47) GPBAR1
SCHEMBL14906396 0.84 GPBAR1 (0.47) GPBAR1
SCHEMBL14895848 0.84 S1PR1 (0.37) GPBAR1NPC1RAB9AHSP90AA1HSP90AB1
SCHEMBL14906387 0.82 GPBAR1 (0.40) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013062887-A1 SUBSTITUTED PYRIDINE DERIVATIVES USEFUL AS GPR131 AGONISTS MERCK SHARP & DOHME CORP. (US) 2013-05-02 WO disclosed