SCHEMBL14907708

SCHEMBL14907708

N=C(NCc1ccnc2[nH]ccc12)Oc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.43
RET P07949 2/20 0.43
JAK2 O60674 2/20 0.43
AURKB Q96GD4 2/20 0.43
IKBKB O14920 1/20 0.43
CHUK O15111 1/20 0.43
DAPK3 O43293 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
PAK4 O96013 1/20 0.43
CSF1R P07333 1/20 0.43
IGF1R P08069 1/20 0.43
FGFR1 P11362 1/20 0.43
PRKACA P17612 1/20 0.43
FLT1 P17948 1/20 0.43
LTK P29376 1/20 0.43
GRK5 P34947 1/20 0.43
KDR P35968 1/20 0.43
MAP2K2 P36507 1/20 0.43
MAPK8 P45983 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14907695 0.79 JAK2 (0.38) ROCK1RETJAK2AURKBIKBKB
SCHEMBL14907704 0.78 MET (0.38) ROCK1RETJAK2AURKBIKBKB
SCHEMBL16141576 0.78 PTK2 (0.38) ROCK1RETJAK2AURKBIKBKB
Hydrochloric Acid SCHEMBL538973 0.76 PRKCI (0.42) ROCK1RETJAK2AURKBIKBKB
SCHEMBL4974852 0.71 NUDT1 (0.41) ROCK1RETJAK2AURKBIKBKB
SCHEMBL4974854 0.71 NUDT1 (0.41) ROCK1RETJAK2AURKBIKBKB
SCHEMBL14907662 0.70 NUDT1 (0.44) ROCK1RETJAK2AURKBIKBKB
SCHEMBL14894258 0.70 JAK2 (0.40) ROCK1RETJAK2AURKBIKBKB
SCHEMBL14907843 0.70 IKBKB (0.40) ROCK1RETJAK2AURKBIKBKB
SCHEMBL14894261 0.70 MEN1 (0.51) JAK2PRKCIAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013062945-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2013-05-02 WO disclosed