SCHEMBL14909183

SCHEMBL14909183

CC(C)(C)N(C(=O)O)c1ccnc(Cl)c1F

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ASPH Q12797 2/20 0.39
KDM8 Q8N371 2/20 0.39
GPBAR1 Q8TDU6 1/20 0.37
ATR Q13535 1/20 0.35
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CNR2 P34972 1/20 0.32
POLB P06746 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
KMO O15229 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
NAPRT Q6XQN6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1350020 0.81 ATR (0.34) KDM4EASPHKDM8ATRLMNA
SCHEMBL238763 0.78 SMN1; SMN2 (0.46) KDM4ELMNASMN1; SMN2POLBTDP1
SCHEMBL6705128 0.77 ATR (0.32) ATRLMNASMN1; SMN2POLBTDP1
SCHEMBL25396869 0.76 NOTUM (0.38) KMO
SCHEMBL1699332 0.75 ATR (0.36) KDM4EASPHKDM8ATRLMNA
SCHEMBL28906545 0.75 SMN1; SMN2 (0.41) KDM4ELMNASMN1; SMN2POLB
SCHEMBL14909869 0.73 PIK3CA (0.40) KDM4EASPHKDM8LMNASMN1; SMN2
SCHEMBL16776759 0.73 GCK (0.39)
SCHEMBL31352713 0.72 SSTR4 (0.41) KDM4EGPBAR1ATRLMNASMN1; SMN2
SCHEMBL28906476 0.72 KEAP1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4737450-A1 HETEROAROMATIC FORMAMIDE COMPOUNDS AND USES THEREOF IN MEDICINE Longwood Pharmaceuticals (Hangzhou) Co., Ltd (CN) 2026-05-06 EP disclosed
WO-2023098425-A1 KRAS INHIBITORS, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 上海和誉生物医药科技有限公司 2023-06-08 WO disclosed
WO-2023098426-A1 7-(NAPHTHALENE-L-YL)PYRIDO[4,3-D]PYRIMIDINE DERIVATIVES, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海和誉生物医药科技有限公司 2023-06-08 WO disclosed
WO-2022161489-A1 PENTAHETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海艾力斯医药科技股份有限公司 2022-08-04 WO disclosed
EP-2589592-B1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM CORP (JP) 2018-08-22 EP disclosed
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-8772320-B2 2014-07-08 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed
EP-2589592-A1 NOVEL NICOTINAMIDE DERIVATIVES OR SALTS THEREOF FUJIFILM Corporation (JP) 2013-05-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK KDM4E 2420/4885ASPH 2422/4885KDM8 1066/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.