SCHEMBL1699332

SCHEMBL1699332

Cc1ccnc(Cl)c1N(C(=O)O)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ASPH Q12797 1/20 0.34
KDM8 Q8N371 1/20 0.34
CNR2 P34972 1/20 0.33
KMO O15229 1/20 0.32
FFAR1 O14842 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
GRM5 P41594 1/20 0.30
RECQL P46063 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
KDM5A P29375 1/20 0.30
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL236945 0.83 CCR1 (0.34) ATRSMN1; SMN2LMNAKDM4EASPH
SCHEMBL23854582 0.79 KDM5A (0.35) ATRKDM4EASPHKDM8KDM5A
SCHEMBL8802786 0.75 ALDH1A1 (0.38) LMNAKDM4EALDH1A1NPSR1
SCHEMBL14909183 0.75 KDM4E (0.39) ATRSMN1; SMN2LMNAKDM4EASPH
SCHEMBL238763 0.74 SMN1; SMN2 (0.46) SMN1; SMN2LMNAKDM4ETDP1ALDH1A1
SCHEMBL1350020 0.74 ATR (0.34) ATRSMN1; SMN2LMNAKDM4EASPH
SCHEMBL1094625 0.71 L3MBTL1 (0.42) SMN1; SMN2LMNACNR2KMOALDH1A1
SCHEMBL71090 0.71 SMARCA2 (0.41) ATRKDM4ECNR2FFAR1ALDH1A1
SCHEMBL6705128 0.71 ATR (0.32) ATRSMN1; SMN2LMNAFFAR1TDP1
SCHEMBL7410941 0.70 HTT (0.45) LMNAKDM4EALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed