SCHEMBL14910052

SCHEMBL14910052

O=[N+]([O-])CCC(O)c1ccc(F)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
ALDH1A1 P00352 2/20 0.39
ADRB1 P08588 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRB3 P13945 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
GRM8 O00222 1/20 0.36
GRM6 O15303 1/20 0.36
GRM4 Q14833 1/20 0.36
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
PDPK1 O15530 1/20 0.33
MME P08473 1/20 0.32
ALDH3A1 P30838 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12285406 1.00 CES2 (0.41) CES2CES1ALDH1A1ADRB1ADRA2A
SCHEMBL30371878 1.00 CES2 (0.41) CES2CES1ALDH1A1ADRB1ADRA2A
SCHEMBL2557213 1.00 CES2 (0.41) CES2CES1ALDH1A1ADRB1ADRA2A
SCHEMBL30372083 1.00 CES2 (0.41) CES2CES1ALDH1A1ADRB1ADRA2A
SCHEMBL14910192 0.81 CES2 (0.35) CES2CES1ALDH1A1GRM8GRM6
SCHEMBL12286385 0.81 PDPK1 (0.38) CES2CES1ALDH1A1AKR1C3AKR1C2
SCHEMBL14923622 0.81 CES2 (0.35) CES2CES1ALDH1A1GRM8GRM6
SCHEMBL28980525 0.76 SIGMAR1 (0.36) CES2CES1ALDH1A1GRM8GRM6
SCHEMBL28980526 0.76 SIGMAR1 (0.36) CES2CES1ALDH1A1GRM8GRM6
SCHEMBL24370650 0.75 CES2 (0.44) CES2CES1ADRB1ADRA2AADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2589587-A1 Synthesis of nitrogen substituted cyclopropanes Chemo Ibérica, S.A. (ES) 2013-05-08 EP claimed
CN-115894496-B Preparation method of ticagrelor and intermediate thereof 上海贝美医药科技有限公司 2025-03-21 CN disclosed
CN-115894496-A Preparation method of ticagrelor and intermediate thereof 上海贝美医药科技有限公司 2023-04-04 CN disclosed
EP-2589587-A1 Synthesis of nitrogen substituted cyclopropanes Chemo Ibérica, S.A. (ES) 2013-05-08 EP disclosed
EP-2589587-A1 Synthesis of nitrogen substituted cyclopropanes Chemo Ibérica, S.A. (ES) 2013-05-08 EP disclosed