SCHEMBL14915166

SCHEMBL14915166

COC=C1C[C@@H](C(=O)OC)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.49
NR1H2 P55055 2/20 0.39
NR1H3 Q13133 1/20 0.39
NPC1 O15118 1/20 0.37
MMP2 P08253 1/20 0.35
ANPEP P15144 1/20 0.35
CYP19A1 P11511 1/20 0.35
PDE4B Q07343 1/20 0.34
HDAC8 Q9BY41 2/20 0.34
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
IMPDH2 P12268 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14915162 1.00 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL21845196 1.00 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL14915165 1.00 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL2380961 0.89 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL2836619 0.89 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL2380958 0.89 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL30987621 0.89 PTPN1 (0.49) PTPN1NR1H2NR1H3NPC1MMP2
SCHEMBL24421263 0.88 NR1H2 (0.42) PTPN1NR1H2NR1H3NPC1PDE4B
SCHEMBL29257431 0.88 NR1H2 (0.42) PTPN1NR1H2NR1H3NPC1PDE4B
SCHEMBL31239774 0.87 PTPN1 (0.48) PTPN1NR1H2NR1H3NPC1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3853234-B1 FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATASE INHIBITORS NIKANG THERAPEUTICS INC (US) 2025-04-23 EP disclosed
US-12264167-B2 Fused tricyclic ring derivatives as SRC homology-2 phosphate inhibitors NIKANG THERAPEUTICS, INC. (US) 2025-04-01 US disclosed
CN-112996795-B Fused tricyclic derivatives as SRC homo-2 phosphatase inhibitors 尼坎治疗公司 2024-11-12 CN disclosed
US-20230167134-A1 FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE INHIBITORS NIKANG THERAPEUTICS, INC. 2023-06-01 US disclosed
US-20230167134-A1 FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE INHIBITORS NIKANG THERAPEUTICS, INC. 2023-06-01 US disclosed
US-11518772-B2 Fused tricyclic ring derivatives as Src homology-2 phosphate inhibitors NIKANG THERAPEUTICS, INC. (US) 2022-12-06 US disclosed
EP-2773634-B1 ROD-LIKE HEPATITIS C VIRUS INHIBITORS CONTAINING THE FRAGEMENT {2-[4-(BIPHENYL-4-YL)-1H-IMIDAZO-2-YL]PYRROLIDINE-1-CARBONLYMETHYL}AMINE THERAVANCE BIOPHARMA R&D IP LLC (US) 2018-06-06 EP disclosed
US-9669027-B2 Hepatitis C virus inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2017-06-06 US disclosed
US-20160038483-A1 HEPATITIS C VIRUS INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC (US) 2016-02-11 US disclosed
US-9212168-B2 Hepatitis C virus inhibitors THERAVANCE BIOPHARMA R&D IP, LLC (US) 2015-12-15 US disclosed
US-20130115194-A1 HEPATITIS C VIRUS INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130115194-A1 HEPATITIS C VIRUS INHIBITORS HAVCR2, SLC10A1, HDGF PTPN1 1088/4885NR1H2 517/4885NR1H3 309/4885
US-20230167134-A1 FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE INHIBITORS SRC, PTPRCAP, PTPRC PTPN1 9/4885NR1H2 2154/4885NR1H3 2503/4885
US-20160038483-A1 HEPATITIS C VIRUS INHIBITORS HAVCR2, SLC10A1, HDGF PTPN1 1088/4885NR1H2 517/4885NR1H3 309/4885
US-12264167-B2 Fused tricyclic ring derivatives as SRC homology-2 phosphate inhibitors SRC, PTPRCAP, PTPRC PTPN1 9/4885NR1H2 2154/4885NR1H3 2503/4885
US-11518772-B2 Fused tricyclic ring derivatives as Src homology-2 phosphate inhibitors SRC, PTPRCAP, PTPRC PTPN1 9/4885NR1H2 2154/4885NR1H3 2503/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.