SCHEMBL14918154

SCHEMBL14918154

FC(F)(F)c1nc(-c2cnc(N3CCNCC3)nc2)no1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 15/20 0.54
HDAC1 Q13547 10/20 0.54
HDAC8 Q9BY41 4/20 0.50
HDAC4 P56524 12/20 0.45
ADRB1 P08588 1/20 0.44
PLAT P00750 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL14918037 0.92 HDAC6 (0.48) HDAC6HDAC1HDAC8HDAC4
SCHEMBL14918111 0.84 HDAC6 (0.63) HDAC6HDAC1HDAC8
SCHEMBL14917670 0.82 HDAC6 (0.53) HDAC6HDAC1HDAC8HDAC4
SCHEMBL14918456 0.80 HDAC4 (0.55) HDAC6HDAC1HDAC8HDAC4
SCHEMBL14917969 0.79 HDAC6 (0.50) HDAC6HDAC1HDAC8HDAC4
SCHEMBL12069976 0.78 ADRB1 (0.46) HDAC6HDAC1HDAC8HDAC4ADRB1
SCHEMBL14918373 0.76 HDAC4 (0.55) HDAC6HDAC1HDAC8HDAC4
SCHEMBL14918477 0.76 HDAC4 (0.70) HDAC6HDAC8HDAC4
SCHEMBL14918156 0.75 SMN1; SMN2 (0.53) HDAC6HDAC1HDAC8HDAC4
SCHEMBL14932826 0.75 HDAC4 (0.68) HDAC6HDAC1HDAC8HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013066831-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO disclosed
WO-2013066831-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2013-05-10 WO disclosed