SCHEMBL14922265

SCHEMBL14922265

CC(=O)COc1ccc(N2CCNCC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.57
HTR3E A5X5Y0 2/20 0.57
HTR3B O95264 2/20 0.57
HTR3A P46098 2/20 0.57
HTR3D Q70Z44 2/20 0.57
HTR3C Q8WXA8 2/20 0.57
SIGMAR1 Q99720 2/20 0.57
TPSAB1 Q15661 1/20 0.51
TPSD1 Q9BZJ3 1/20 0.51
TPSG1 Q9NRR2 1/20 0.51
LTA4H P09960 4/20 0.50
MAPK1 P28482 2/20 0.48
USP2 O75604 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
MAPT P10636 3/20 0.46
GAA P10253 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12814351 0.86 ITGB3 (0.62) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL14922325 0.83 MEN1 (0.55) MAPK1TSHRHSD17B10ITGB3ITGA2B
SCHEMBL12814058 0.83 NPSR1 (0.58) ADRB1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL12814057 0.82 NPSR1 (0.57) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7366682 0.82 ADRB1 (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8325106 0.80 ITGB3 (0.55) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL4543250 0.80 ADRB1 (0.62) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8662762 0.79 ITGB3 (0.54) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL8662766 0.79 ITGB3 (0.54) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2155052 0.79 ADRB1 (0.66) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed