SCHEMBL14922285

SCHEMBL14922285

CN1CCN(c2ccc(F)cc2C#N)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
XDH P47989 1/20 0.45
ROCK2 O75116 2/20 0.45
ROCK1 Q13464 2/20 0.45
CDC42BPB Q9Y5S2 2/20 0.45
GAA P10253 2/20 0.43
LMNA P02545 1/20 0.43
KDM4E B2RXH2 4/20 0.43
TSHR P16473 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29817937 0.89 ALDH1A1 (0.55) ALDH1A1L3MBTL1HTR3EHTR3BHTR3A
SCHEMBL13419452 0.81 KDM4E (0.57) ALDH1A1HTR3AXDHROCK2ROCK1
SCHEMBL29703766 0.80 MAPT (0.63) ALDH1A1L3MBTL1XDHROCK2ROCK1
SCHEMBL2997329 0.80 ALDH1A1 (0.57) ALDH1A1HTR3AROCK2ROCK1CDC42BPB
SCHEMBL431886 0.80 DRD4 (0.48) ALDH1A1L3MBTL1XDHROCK2ROCK1
SCHEMBL24518337 0.80 XDH (0.45) ALDH1A1L3MBTL1XDHROCK2ROCK1
SCHEMBL24309700 0.80 XDH (0.48) ALDH1A1L3MBTL1XDHROCK2ROCK1
SCHEMBL5654064 0.80 MAPT (0.63) ALDH1A1L3MBTL1XDHROCK2ROCK1
SCHEMBL1484007 0.80 POLB (0.61) ALDH1A1HTR3AXDHROCK2ROCK1
SCHEMBL3578305 0.80 MAPK1 (0.55) ALDH1A1L3MBTL1XDHROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed