SCHEMBL14922299

SCHEMBL14922299

CC(C)OCCOc1ccc(N2CCN(C)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.56
MAPT P10636 3/20 0.52
HPGD P15428 3/20 0.52
TSHR P16473 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
KCNH2 Q12809 1/20 0.47
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
ADRA2C P18825 1/20 0.45
GFER P55789 1/20 0.45
PTK2B Q14289 1/20 0.45
ESR2 Q92731 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
HTR1A P08908 5/20 0.44
HTR1D P28221 1/20 0.44
HTR1B P28222 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14922263 0.84 ADRB1 (0.55) HRH3HPGDKCNH2HTR1AHTR1D
SCHEMBL8275460 0.83 HRH3 (0.59) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL22022308 0.81 HRH3 (0.61) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL14922313 0.80 HRH3 (0.57) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL16218812 0.80 DRD2 (0.59) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL21659428 0.80 HRH3 (0.68) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL14922320 0.80 HRH3 (0.52) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL8363114 0.80 HRH3 (0.63) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL14922311 0.79 HRH3 (0.56) HRH3MAPTHPGDTSHRTAAR1
SCHEMBL21659290 0.78 HRH3 (0.79) HRH3MAPTHPGDKCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed