SCHEMBL14922338

SCHEMBL14922338

CC(C)C(=O)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CTSK P43235 6/20 0.39
CTSS P25774 2/20 0.39
CA12 O43570 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CYP2D6 P10635 1/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
TRPA1 O75762 1/20 0.36
AAK1 Q2M2I8 2/20 0.36
APLNR P35414 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
DGAT1 O75907 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
PREP P48147 1/20 0.34
NFKB1 P19838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL890057 0.83 POLB (0.30) CA12CA14
SCHEMBL14276786 0.78 TDP1 (0.39) CA1CA2CA7CTSKCA12
SCHEMBL16391154 0.77 TDP1 (0.42) CA1CA2CA7CTSKCTSS
SCHEMBL16391151 0.77 TDP1 (0.42) CA1CA2CA7CTSKCTSS
SCHEMBL15113634 0.77 CA1 (0.41) CA1CA2CA7CTSKCTSS
SCHEMBL17712226 0.76 CA1 (0.40) CA1CA2CA7CTSKCTSS
SCHEMBL7922248 0.76 PIK3CD (0.47) CA1CA2CA7CTSKCTSS
SCHEMBL76832 0.76 KDM4C (0.41) CA1CA2CA7CTSKCTSS
SCHEMBL9304597 0.74 APLNR (0.38) CA1CA2CA7CTSKCTSS
SCHEMBL21834933 0.74 KDM4C (0.39) CA1CA2CA7CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed