SCHEMBL9304597

SCHEMBL9304597

CC(C)(C)OC(=O)NC(C)(C)C(=O)F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
DGAT1 O75907 1/20 0.37
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 3/20 0.34
CA14 Q9ULX7 3/20 0.34
CTSK P43235 3/20 0.34
CTSS P25774 1/20 0.34
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14276786 0.81 TDP1 (0.39) APLNRTDP1DGAT1CA1CA2
SCHEMBL28918296 0.81 APLNR (0.40) APLNRTDP1DGAT1CA1CA2
SCHEMBL76832 0.79 KDM4C (0.41) APLNRTDP1DGAT1CA1CA2
SCHEMBL1374814 0.77 DGAT1 (0.52) APLNRTDP1DGAT1CA1CA2
SCHEMBL21952155 0.77 TDP1 (0.37) APLNRTDP1DGAT1CA1CA2
SCHEMBL20295137 0.77 GAA (0.39) APLNRTDP1DGAT1CA1CA2
SCHEMBL7771576 0.77 TDP1 (0.37) APLNRTDP1DGAT1CA1CA2
SCHEMBL21834933 0.77 KDM4C (0.39) APLNRTDP1DGAT1CA1CA2
SCHEMBL19154278 0.77 TDP1 (0.37) APLNRTDP1DGAT1CA1CA2
SCHEMBL4197524 0.77 TDP1 (0.37) APLNRTDP1DGAT1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085429-B Aromatic heterocyclic derivative and application thereof in medicines 广东东阳光药业有限公司 2019-12-10 CN disclosed
EP-0495265-B1 Acid-labile linker molecules AKZO NOBEL NV (NL) 1994-08-03 EP disclosed
US-5306809-A Cancer immune therapy AKZO N.V. (NL) 1994-04-26 US disclosed
EP-0495265-A1 Acid-labile linker molecules Akzo Nobel N.V. (NL) 1992-07-22 EP disclosed