SCHEMBL14922720

SCHEMBL14922720

COc1c(Cl)cc(N2CCN(C)CC2)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.56
DRD4 P21917 3/20 0.56
DRD3 P35462 3/20 0.56
HTR1A P08908 2/20 0.56
HTR2A P28223 2/20 0.56
HTR2C P28335 2/20 0.56
HRH4 Q9H3N8 1/20 0.46
BRD4 O60885 1/20 0.43
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
RAD52 P43351 1/20 0.41
SIRT6 Q8N6T7 1/20 0.41
HTR6 P50406 1/20 0.41
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41
ADRA2C P18825 2/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5245685 0.80 ADRB1 (0.61) DRD2DRD4DRD3HTR1AHTR2A
Hydrochloric Acid SCHEMBL4934648 0.79 ADRB1 (0.59) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL23657292 0.75 ADRB1 (0.58) DRD2DRD3HRH4DRD1DRD5
SCHEMBL8318081 0.74 BCL2A1 (0.59) MAPTKDM4ESIRT6ADRA2CALDH1A1
SCHEMBL423400 0.73 MAPT (0.65) DRD2DRD4DRD3DRD1DRD5
SCHEMBL14922319 0.73 CHKA (0.46) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL24309441 0.73 SIRT6 (0.45) DRD2DRD3HRH4MAPTKDM4E
SCHEMBL8318825 0.72 MAPT (0.59) L3MBTL1MAPTKDM4EADRA2CALDH1A1
SCHEMBL24309440 0.72 CCR1 (0.40) DRD2DRD4DRD3HTR1AHTR2A
SCHEMBL24309761 0.71 SIRT6 (0.44) HRH4MAPTKDM4ERAD52SIRT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44205-E1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. (US) 2013-05-07 US disclosed