SCHEMBL14923264

SCHEMBL14923264

CC(C)CC1(C)C(=O)N(CCC2CCN(C(=O)C(C)c3ccccc3)CC2)C(=N)N1C

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 10/20 0.43
GAA P10253 2/20 0.40
RAB9A P51151 1/20 0.39
CHRM3 P20309 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CNR1 P21554 2/20 0.37
CNR2 P34972 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520697 0.83 TRPV1 (0.41) TRPV1GAARAB9ACHRM3ALDH1A1
SCHEMBL7528142 0.77 ADAMTS5 (0.40) TRPV1GAARAB9ACHRM3ALDH1A1
SCHEMBL7522013 0.76 ADAMTS5 (0.42) TRPV1GAACNR1CNR2GPR55
SCHEMBL8265223 0.74 BACE1 (0.33) ALDH1A1
SCHEMBL7521184 0.71 HDAC3 (0.42) ALDH1A1
SCHEMBL13475756 0.71 ADAMTS5 (0.40) TRPV1GAARAB9AALDH1A1CNR1
SCHEMBL17551041 0.70 BACE1 (0.35) CNR1CNR2
SCHEMBL7520459 0.70 KMT2A (0.46) GAAALDH1A1
SCHEMBL7522535 0.70 CHRM3 (0.39) TRPV1RAB9ACHRM3ALDH1A1CNR1
SCHEMBL7519913 0.70 TRPV1 (0.35) TRPV1GAARAB9ACHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699455-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2013-05-08 EP disclosed