SCHEMBL14923400

SCHEMBL14923400

CCCN[C@H]1CCC[C@@H](CNC(=N)N(C)C(=O)CCC2CCCCC2)C1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.36
EPHX1 P07099 12/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31
S1PR5 Q9H228 1/20 0.31
EPHX2 P34913 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14923323 1.00 HPGD (0.36) HPGDEPHX1ALDH1A1KDM4EMEN1
SCHEMBL14923325 0.92 HPGD (0.36) HPGDEPHX1MEN1KMT2ANPC1
SCHEMBL17715619 0.89 CTSD (0.38) HPGDEPHX1KDM4EMEN1KMT2A
SCHEMBL14923346 0.87 HPGD (0.39) HPGDEPHX1MEN1KMT2ANPC1
SCHEMBL14923302 0.87 HPGD (0.39) HPGDEPHX1MEN1KMT2ANPC1
SCHEMBL14923324 0.85 HPGD (0.34) HPGDEPHX1ALDH1A1MEN1KMT2A
SCHEMBL14923374 0.83 EPHX1 (0.42) HPGDEPHX1ALDH1A1MEN1KMT2A
SCHEMBL17715611 0.82 HTR5A (0.43) HPGDEPHX1ALDH1A1KMT2ANPC1
SCHEMBL14923312 0.82 HPGD (0.35) HPGDEPHX1ALDH1A1MEN1KMT2A
SCHEMBL17551587 0.81 HPGD (0.34) HPGDEPHX1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343069-B1 Heterocyclic aspartyl protease inhibitors MERCK SHARP & DOHME (US) 2016-03-02 EP disclosed
EP-1699455-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2013-05-08 EP disclosed