SCHEMBL14928818

SCHEMBL14928818

C[C@H](CN1C(=O)c2ccccc2C1=O)c1ccsc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
TDP1 Q9NUW8 1/20 0.40
KMT2A Q03164 3/20 0.39
CASP3 P42574 2/20 0.39
POLB P06746 1/20 0.37
MAOB P27338 2/20 0.37
MAPK1 P28482 1/20 0.37
ELANE P08246 1/20 0.37
PKM P14618 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
GLS O94925 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14923682 0.82 ALDH1A1 (0.41) ALDH1A1KMT2ACASP3MAPK1ELANE
SCHEMBL10722361 0.80 KMT2A (0.50) ALDH1A1TDP1KMT2ACASP3MAPK1
SCHEMBL6556286 0.80 KMT2A (0.50) ALDH1A1TDP1KMT2ACASP3MAPK1
SCHEMBL14928651 0.80 KMT2A (0.50) ALDH1A1TDP1KMT2ACASP3MAPK1
SCHEMBL111864 0.78 ALDH1A1 (0.42) ALDH1A1KMT2APOLB
SCHEMBL14911465 0.75 ALDH1A1 (0.42) ALDH1A1KMT2AMAPK1CA12CA9
SCHEMBL2564111 0.75 CASP3 (0.53) ALDH1A1KMT2ACASP3POLBPKM
SCHEMBL2564113 0.75 CASP3 (0.53) ALDH1A1KMT2ACASP3POLBPKM
SCHEMBL14910738 0.73 KMT2A (0.43) ALDH1A1KMT2ACASP3POLBMAOB
SCHEMBL14910736 0.73 KMT2A (0.43) ALDH1A1KMT2ACASP3POLBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895585-B2 Nicotinamide derivative or salt thereof FUJIFILM CORPORATION (JP) 2014-11-25 US disclosed
US-8809371-B2 2014-08-19 US disclosed
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK ALDH1A1 1638/4885TDP1 2598/4885KMT2A 1162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.